RU58841 masana'antar foda Lambar CAS: 154992-24-2 Tsarkakakken 99.0% min. don ƙarin sinadaran
Sigogin Samfura
| Sunan samfurin | 4-[3-(4-Hydroxybutyl)-4,4-dimethyl-2,5-dioxo-1-imidazolidinyl]-2-(trifluoromethyl)benzonitrile |
| Wani suna | RU58841 |
| Lambar CAS | 154992-24-2 |
| Tsarin kwayoyin halitta | C17H18F3N3O3 |
| Nauyin kwayoyin halitta | 369.34 |
| Tsarkaka | 99.0% |
| Bayyanar | farin foda |
| shiryawa | 1kg/jaka |
| Aikace-aikace | Gashi mai sheƙi |
Gabatarwar samfur
RU58841 (wanda aka fi sani da RU-58841) wani sinadari ne, RU58841 yana fafatawa da dihydrotestosterone don kiyaye matakan DHT a cikin matsakaicin yanayi, ta haka yana daidaita zagayowar girman gashi. Yana ƙarfafa canza sabbin gashin gashi zuwa gashin anagen ta hanyar shiga matakin anagen. Barin gashin da suka lalace lokaci ya koma matakin girma na yau da kullun yana taimaka wa ƙwayoyin halitta su murmure. Hakanan yana ƙara kwararar jini zuwa ga gashin da suka lalace kuma yana taimaka musu su sake farfaɗowa. A gefe guda kuma, RU58841 (RU-58841) yana aiki ta hanyar ɗaurewa ga masu karɓar androgen a cikin gashin. Don haka androgens ba su da damar ɗaurewa da fara amsawar sarkar na alopecia na androgenetic da fara aikin da ake kira miniaturization. An nuna yana katse wannan saƙon asarar gashi a gida don ci gaba da haɓakar gashi na yau da kullun.
Fasali
(1) Zai iya hana asarar gashi: RU58841 wani magani ne na musamman da ke hana samar da hormone, wanda zai iya hana haɗakar ƙwayoyin halittar gashi na androgen da fatar kai, ta haka ne zai rage haɗarin asarar gashi.
(2) Sha mai kyau: RU58841 yana da ƙaramin nauyin ƙwayoyin halitta, tsari mai sauƙi, kuma yana da sauƙin sha. Yana iya shiga jiki da sauri kuma ya fara aiki cikin ɗan gajeren lokaci.
(3) Babban zaɓi ga androgen: RU58841 zai iya hana aikin androgen ba tare da shafar wasu hormones ba.
(4) Tsawon lokacin aiki: RU58841 yana da tsawon rabin rai a jiki, yana iya ci gaba da hana tasirin androgen, kuma tsawon lokacin tasirin na iya zama har zuwa awanni 48.
(5) Tsarkakakken abu: Ta hanyar cirewa ta halitta da kuma tsarin kera kayayyaki masu kyau, ci gaban RU58841 na iya samun samfuran tsafta mai yawa.
Aikace-aikace
A cikin bincike da gwaje-gwajen asibiti, an nuna cewa RU58841 yana ƙara yawan kwafi na ƙwayoyin halitta a cikin ƙwayoyin stromal, yana ƙara yawan ƙwayoyin halitta a cikin ƙwayoyin tushe na waje da kuma ƙara girman gashi da yawan gashi, don haka RU58841 magani ne na bincike don maganin alopecia na androgenetic. Babban ƙa'idar aiki ita ce toshe haɗin DHT da AR na ƙwayoyin gashi, wanda galibi ana amfani da shi don magance matsalolin asarar gashi da asarar gashi.












