Mai ƙera foda na CMS121 Lambar CAS: 1353224-53-9 Tsarkakakken kashi 98.0% na mintuna don ƙarin sinadaran
Sigogin Samfura
| Sunan samfurin | CMS121 |
| Wani suna | CMS-121; 1,2-Benzenediol,4-[4-(cyclopentyloxy)-2-quinolinyl]-; 4-(4-(cyclopentyloxy)quinolin-2-yl)benzene-1,2-diol(CMS121); ACC,AcetylCoenzymeACarboxylase,cuta,neuroprotective,inhibit,anti-inflammatory,mitochondria,Alzheimer's,antioxidative,acetylation,Inhibitor,H3K9,Acetyl-CoACarboxylase,CMS121,dementia,ACC1,CMS-121 |
| Lambar CAS | 1353224-53-9 |
| Tsarin kwayoyin halitta | C20H19NO3 |
| Nauyin kwayoyin halitta | 321.37 |
| Tsarkaka | 98.0% |
| Bayyanar | Foda mai launin rawaya mai haske |
| Aikace-aikace | Kayan Abinci Mai Gina Jiki |
Gabatarwar samfur
4-(4-(cyclopentyloxy)quinolin-2-yl)benzene-1,2-diol wani sinadari ne wanda kuma ake kira CMS121. Tsarin sinadari yana nuna cewa yana da siffofi na musamman da kuma amfani mai yuwuwa. Don fahimtar muhimmancinsa, yana taimakawa wajen gano ƙungiyoyin aiki da ke akwai da kuma nazarin tasirinsu. Kasancewar zoben quinoline yana nuna cewa sinadari na iya aiki a fannin ilmin halitta. An san ƙwayoyin da Quinoline ya samo asali saboda nau'ikan sinadari daban-daban, gami da ayyukan kashe ƙwayoyin cuta da hana kumburi. Haɗa ƙungiyar cyclopentyloxy na iya taimakawa wajen narkewar sinadari ko kuma haɓaka aikinsa na halitta ta hanyar tasirin steric. A cikin bincike kan ƙwayoyin HT22, CMS-121 ya nuna tasirin kariya daga jijiyoyi masu mahimmanci, yana kare waɗannan ƙwayoyin daga ischemia da lalacewar oxidative. Bugu da ƙari, CMS-121 yana da manyan sifofin hana kumburi, yana nuna ikonsa na daidaita martanin kumburi. Ta hanyar yin hakan, CMS-121 yana da yuwuwar rage kumburi a cikin kyallen takarda da gabobin jiki daban-daban. CMS-121 yana da ƙarfin aikin magunguna a matsayin mai hana acetyl-CoA carboxylase 1 (ACC1). Ƙarfin tasirinsa na hana ACC1 yana sa ya zama wani abu mai kyau.
Fasali
(1) Tsafta mai yawa: CMS-121 na iya samun samfuran tsafta mai yawa ta hanyar ingantattun hanyoyin samarwa. Tsafta mai yawa yana nufin ingantaccen samuwar halittu da ƙarancin halayen da ba su da kyau.
(2) Tsaro: Babban aminci, ƙarancin halayen da ba su dace ba.
(3) Kwanciyar hankali: CMS-121 yana da kyakkyawan kwanciyar hankali kuma yana iya kiyaye aikinsa da tasirinsa a ƙarƙashin yanayi daban-daban da yanayin ajiya.
Aikace-aikace
CMS-121 wani maganin quinolone ne kuma maganin acetyl-CoA carboxylase 1 (ACC1) mai aiki ta baki wanda ke da kyawawan halaye na magani. An gudanar da bincike mai zurfi don bincika fa'idodin CMS-121 a fannoni daban-daban, ciki har da kariyar jijiyoyi, tasirin hana kumburi, aikin antioxidant, da tasirinsa akan alamun da ke da alaƙa da tsufa mai lafiya.












