Mai ƙera foda na Nefiracetam CAS No.: 77191-36-7 Tsarkakakken kashi 99% na minti ɗaya don ƙarin sinadaran
Bidiyon Samfuri
Sigogin Samfura
| Sunan samfurin | Nefiracetam |
| Wani suna | n-(2,6-dimethylphenyl)-2-oxo-1-pyrrolidineacetamide;NEFIRACETAM; 2-oxo-1-pyrrolidinylaseticacid,2,6-dimethylanilide; dm9384; n-(2,6-dimethylphenyl)-2-oxo-1-pyrrolidineacetamid;DM-9384,(2-(2-Oxopyrrolidin-1-yl)-N-(2,6-dimethylphenyl)-acetamide); DMMPA |
| Lambar CAS | 77191-36-7 |
| Tsarin kwayoyin halitta | C14H18N2O2 |
| Nauyin kwayoyin halitta | 246.3 |
| Tsarkaka | 99.0% |
| Bayyanar | Foda fari |
| shiryawa | 25 kg/ganga |
| Aikace-aikace | nootropic |
Gabatarwar samfur
Nefiracetam na cikin dangin piracetam, wani nau'in magunguna da aka sani da halayensu na haɓaka fahimta. An fara haɗa Nefiracetam a farkon shekarun 1980 kuma cikin sauri ya jawo hankali saboda tsarin aikinsa na musamman da kuma yuwuwar amfani da shi wajen warkar da cututtuka. Ana tsammanin wannan sinadarin racemic yana shafar neurotransmitters da receptors a cikin kwakwalwa, wanda a ƙarshe yana haɓaka ingantattun ƙwarewar fahimta. Nefiracetam galibi yana shafar matakan kwakwalwa na acetylcholine, babban mai ba da amsa ga ƙwaƙwalwa wanda ke da alhakin ƙwaƙwalwa, koyo, da aikin fahimta. Ta hanyar daidaita masu karɓar acetylcholine, nefiracetam yana haɓaka haɓaka sadarwa tsakanin ƙwayoyin jijiyoyi, ta haka yana haɓaka ƙarfin synaptic da inganta riƙewar ƙwaƙwalwa. Bugu da ƙari, nefiracetam yana hulɗa da masu karɓar gamma-aminobutyric acid (GABA) don taimakawa wajen daidaita yanayin neurotransmitter. Ta hanyar tasiri mai kyau ga masu ba da amsa ga motsin rai da hanawa, nefiracetam yana taimakawa wajen kula da aikin kwakwalwa mafi kyau, ta haka yana inganta mayar da hankali, hankali, da kuma aikin fahimta gabaɗaya.
Fasali
(1) Tsafta mai yawa: Nefiracetam na iya samun samfuran tsafta mai yawa ta hanyar tace hanyoyin samar da kayayyaki. Tsafta mai yawa yana nufin ingantaccen samuwar halittu da ƙarancin halayen da ba su da kyau.
(2) Tsaro: Babban aminci, ƙarancin halayen da ba su dace ba.
(3) Kwanciyar hankali: Nefiracetam yana da kyakkyawan kwanciyar hankali kuma yana iya kiyaye aikinsa da tasirinsa a ƙarƙashin yanayi daban-daban da yanayin ajiya.
Aikace-aikace
Nefiracetam wani sinadari ne da aka samo daga piracetam wanda ke hana ruwa shiga jiki, wanda galibi ana ɗaukarsa a matsayin wani sinadari da ke da alhakin gano hanyoyin calcium a cikin jiki da kuma canja wurin abubuwan siginar da ke motsa jiki kai tsaye a matsayin wani ɓangare na agonist na tashoshin calcium ion. Wurin ɗaure Glycine na mai karɓar NDMA. Ta hanyar tasirinsa akan kwakwalwa ta kwakwalwa, nefiracetam na iya haɓaka ƙwarewar fahimta da hana lalacewar koyo da ƙwaƙwalwa. Ba ya da agonist na mai karɓar muscarinic ko halayen antagonist, kuma baya hana aikin acetylcholinease. Saboda haka, tasirinsa na hana amnestic da haɓaka ƙwaƙwalwa ana samun su ta hanyar inganta sakin acetylcholine a cikin kwakwalwa ta kwakwalwa.












